Ian Gilbert IanGilbert,ProfessorofUniversityofDundee,Dundee,U.K.Heisamedicinalchemistandmyresearchinterestsareinthedesignandsynthesisofpotentialdrugs.ThemainstayofhisworkissyntheticmedicinalchemistryaspartoftheDrugDiscoveryUnit(DDU).Wherepossiblehemakeextensiveuseofmolecularmodelingtoguideoursyntheticefforts.Ihaveaparticularinterestsinthefollowingaspectsofdrugdiscovery:NeglecteddiseasessuchashumanAfricantrypanosomiasis,leishmaniasisandmalaria.Chemicalvalidationofdrugtargets,includingnoveltargetsforwhichthereislittleornoprecedencefordrugdiscovery.Novelapproachestoandparadigmsfordrugdiscovery.Modeofactionstudiesandtargetidentification.HeisHeadofChemistryintheDDU.Hismainfocusesareonneglecteddiseasesandnoveldrugtargets.Theneglecteddiseaseshearetacklingaremalaria,tuberculosisandthekinetoplastiddiseases.Heusebothtarget-basedapproachesandphenotypicapproaches(wholeparasitescreening).HehavehadparticularsuccessinvalidatingtheenzymeN-myristoyltransferaseasadrugtargetinhumanAfricantrypanosomiasis,andinidentif
IanGilbert,ProfessorofUniversityofDundee,Dundee,U.K.Heisamedicinalchemistandmyresearchinterestsareinthedesignandsynthesisofpotentialdrugs.ThemainstayofhisworkissyntheticmedicinalchemistryaspartoftheDr...
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